β-Carbolines as intermediates in indirect heteroarylation of tryptamines exemplified by the synthesis of 2-pyrazolyltryptamines

β-Carbolines as intermediates in indirect heteroarylation of tryptamines exemplified by the synthesis of 2-pyrazolyltryptamines

A cyclization–recyclization pathway for indirect 2-heteroarylation of tryptamines has been suggested by the example of introducing the pyrazolyl moiety. The process involves the intermediate cyclization of tryptamines into push–pull type β-carboline semi-products. The relative stability of the tauto...

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Главные авторы:	Demidov, O. P., Демидов, О. П.
格式:	Статья
语言:	English
出版:	2023
主题:	1-aroylmethylidene-1,2, 3, 4-tetrahydro-β-carbolines Tryptamines β-carbolines Recyclization Quantum chemical calculations Pyrazolylmelatonins 2-(pyrazol-3-yl)tryptamine 2-(pyrazol-3-yl)-O-methylserotonins
在线阅读:	https://dspace.ncfu.ru/handle/20.500.12258/25810
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