Synthesis of meta-substituted anilines via a three-component reaction of acetone, amines, and 1,3-diketones

Synthesis of meta-substituted anilines via a three-component reaction of acetone, amines, and 1,3-diketones

A facile method for the synthesis of meta-substituted arylamines from acyclic precursors was developed. This method is based on three-component cyclo-condensation/aromatization of in situ generated imines of acetone with 1,3-diketones either under conventional heating or under microwave irradiation....

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Dettagli Bibliografici
Autori principali:	Rubin, M. A., Рубин, М. А.
Natura:	Статья
Lingua:	English
Pubblicazione:	ROYAL SOC CHEMISTRY 2019
Soggetti:	Pd-at-pani Pharmacokinetic properties Trifluoromethyl ketones Pactical catalyst Discovery Inhibitors Potent Benzannulation Condensation Bicalutamide
Accesso online:	http://apps.webofknowledge.com/full_record.do?product=WOS&search_mode=GeneralSearch&qid=1&SID=C2RI3BOJAwOaexjHfEf&page=1&doc=1 https://dspace.ncfu.ru/handle/20.500.12258/9753
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